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David D N'Da
David D N'Da
Verified email at nwu.ac.za - Homepage
Title
Cited by
Cited by
Year
Prodrug strategies for enhancing the percutaneous absorption of drugs
DD N’Da
Molecules 19 (12), 20780-20807, 2014
1292014
Considerations on the mechanism of action of artemisinin antimalarials: Part 1-The'carbon radical'and'heme'hypotheses
R K Haynes, KW Cheu, D N'Da, P Coghi, D Monti
Infectious Disorders-Drug Targets (Formerly Current Drug Targets-Infectious …, 2013
1012013
Synthesis, characterization and antimalarial activity of quinoline–pyrimidine hybrids
SI Pretorius, WJ Breytenbach, C De Kock, PJ Smith, DD N’Da
Bioorganic & medicinal chemistry 21 (1), 269-277, 2013
992013
Recent progress in the development of anti-malarial quinolones
RM Beteck, FJ Smit, RK Haynes, DD N’Da
Malaria journal 13, 1-10, 2014
942014
An update on derivatisation and repurposing of clinical nitrofuran drugs
NH Zuma, J Aucamp, DND David
European Journal of Pharmaceutical Sciences 140, 105092, 2019
712019
Synthesis, in vitro antimalarial activity and cytotoxicity of novel 4-aminoquinolinyl-chalcone amides
FJ Smit, DD N’Da
Bioorganic & Medicinal Chemistry 22 (3), 1128-1138, 2014
682014
Synthesis and in vitro biological evaluation of dihydroartemisinyl-chalcone esters
FJ Smit, RA van Biljon, LM Birkholtz, DND David
European journal of medicinal chemistry 90, 33-44, 2015
592015
Synthesis and in vitro biological evaluation of aminoacridines and artemisinin–acridine hybrids
JP Joubert, FJ Smit, L Du Plessis, PJ Smith, DD N’Da
European Journal of Pharmaceutical Sciences 56, 16-27, 2014
532014
Synthesis and in vitro antimalarial activity of a series of bisquinoline and bispyrrolo [1, 2a] quinoxaline compounds
L Van Heerden, TT Cloete, JW Breytenbach, C de Kock, PJ Smith, ...
European journal of medicinal chemistry 55, 335-345, 2012
522012
Synthesis, in vitro antimalarial and cytotoxicity of artemisinin-aminoquinoline hybrids
MC Lombard, DD N’Da, JC Breytenbach, PJ Smith, CA Lategan
Bioorganic & medicinal chemistry letters 21 (6), 1683-1686, 2011
502011
Synthesis, in vitro antiplasmodial and antiproliferative activities of a series of quinoline–ferrocene hybrids
DD N’Da, PJ Smith
Medicinal Chemistry Research 23, 1214-1224, 2014
492014
Antimalarial and anticancer activities of artemisinin–quinoline hybrid-dimers and pharmacokinetic properties in mice
MC Lombard, DD N’Da, JC Breytenbach, NI Kolesnikova, CT Van Ba, ...
European journal of pharmaceutical sciences 47 (5), 834-841, 2012
452012
Artemisinin–quinoline hybrid-dimers: Synthesis and in vitro antiplasmodial activity
MC Lombard, DD N’Da, JC Breytenbach, PJ Smith, CA Lategan
Bioorganic & medicinal chemistry letters 20 (23), 6975-6977, 2010
442010
Synthesis, in vitro antimalarial activities and cytotoxicities of amino-artemisinin-ferrocene derivatives
C De Lange, D Coertzen, FJ Smit, JF Wentzel, HN Wong, LM Birkholtz, ...
Bioorganic & medicinal chemistry letters 28 (3), 289-292, 2018
412018
Synthesis, in vitro antiplasmodial activity and cytotoxicity of a series of artemisinin–triazine hybrids and hybrid-dimers
TT Cloete, C de Kock, PJ Smith, DND David
European journal of medicinal chemistry 76, 470-481, 2014
342014
Synthesis, antimalarial activities and cytotoxicities of amino-artemisinin-1, 2-disubstituted ferrocene hybrids
C De Lange, D Coertzen, FJ Smit, JF Wentzel, HN Wong, LM Birkholtz, ...
Bioorganic & Medicinal Chemistry Letters 28 (19), 3161-3163, 2018
332018
Accessible and distinct decoquinate derivatives active against Mycobacterium tuberculosis and apicomplexan parasites
RM Beteck, R Seldon, D Coertzen, ME van der Watt, J Reader, ...
Communications Chemistry 1 (1), 62, 2018
332018
Potent in vivo anti-malarial activity and representative snapshot pharmacokinetic evaluation of artemisinin-quinoline hybrids
MC Lombard, DD N’Da, C Tran Van Ba, S Wein, J Norman, L Wiesner, ...
Malaria Journal 12, 1-7, 2013
322013
The cytotoxic activity of macromolecular ferrocene conjugates against the Colo 320 DM human colon cancer line
MT Johnson, E Kreft, DD N'Da, EW Neuse, CEJ van Rensburg
Journal of Inorganic and Organometallic Polymers 13, 255-267, 2003
302003
Recent advances in the synthesis and development of nitroaromatics as anti-infective drugs
C Kannigadu, D N'Da
Current Pharmaceutical Design 26 (36), 4658-4674, 2020
272020
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