| Pharmacology and structure‐activity relationships of bioactive polycyclic cage compounds: a focus on pentacycloundecane derivatives WJ Geldenhuys, SF Malan, JR Bloomquist, AP Marchand, ... Medicinal research reviews 25 (1), 21-48, 2005 | 237 | 2005 |
| Inhibition of monoamine oxidase B by selected benzimidazole and caffeine analogues D van den Berg, KR Zoellner, MO Ogunrombi, SF Malan, G Terre’Blanche, ... Bioorganic & medicinal chemistry 15 (11), 3692-3702, 2007 | 91 | 2007 |
| Synthesis and biological evaluation of pentacyclo [5.4. 0.02, 6.03, 10.05, 9] undecane derivatives as potential therapeutic agents in Parkinson's disease WJ Geldenhuys, SF Malan, T Murugesan, CJ Van der Schyf, ... Bioorganic & medicinal chemistry 12 (7), 1799-1806, 2004 | 82 | 2004 |
| Physicochemical prediction of a brain–blood distribution profile in polycyclic amines J Zah, G Terre'Blanche, E Erasmus, SF Malan Bioorganic & medicinal chemistry 11 (17), 3569-3578, 2003 | 56 | 2003 |
| Thio-and aminocaffeine analogues as inhibitors of human monoamine oxidase HP Booysen, C Moraal, G Terre’Blanche, A Petzer, JJ Bergh, JP Petzer Bioorganic & medicinal chemistry 19 (24), 7507-7518, 2011 | 41 | 2011 |
| Screening of novel pentacyclo-undecylamines for neuroprotective activity WJ Geldenhuys, G Terre'Blanche, CJ Van der Schyf, SF Malan European journal of pharmacology 458 (1-2), 73-79, 2003 | 41 | 2003 |
| 1, 3, 7-Triethyl-substituted xanthines—possess nanomolar affinity for the adenosine A1 receptor MM Van der Walt, G Terre’Blanche Bioorganic & medicinal chemistry 23 (20), 6641-6649, 2015 | 39 | 2015 |
| Structure–activity relationships in the inhibition of monoamine oxidase B by 1-methyl-3-phenylpyrroles MO Ogunrombi, SF Malan, G Terre’Blanche, N Castagnoli Jr, JJ Bergh, ... Bioorganic & medicinal chemistry 16 (5), 2463-2472, 2008 | 37 | 2008 |
| 2-Aminopyrimidines as dual adenosine A1/A2A antagonists SJ Robinson, JP Petzer, G Terre’Blanche, A Petzer, MM Van der Walt, ... European Journal of Medicinal Chemistry 104, 177-188, 2015 | 33 | 2015 |
| The adenosine A2A antagonistic properties of selected C8-substituted xanthines MM Van der Walt, G Terre’Blanche, A Petzer, ACU Lourens, JP Petzer Bioorganic chemistry 49, 49-58, 2013 | 33 | 2013 |
| Inhibition of monoamine oxidase B by N-methyl-2-phenylmaleimides CI Manley-King, G Terre’Blanche, N Castagnoli Jr, JJ Bergh, JP Petzer Bioorganic & medicinal chemistry 17 (8), 3104-3110, 2009 | 29 | 2009 |
| Evaluation of 2‐benzylidene‐1‐tetralone derivatives as antagonists of A1 and A2A adenosine receptors LJ Legoabe, MM Van der Walt, G Terre'Blanche Chemical biology & drug design 91 (1), 234-244, 2018 | 22 | 2018 |
| 5-Substituted 2-benzylidene-1-tetralone analogues as A1 and/or A2A antagonists for the potential treatment of neurological conditions HDJ van Rensburg, G Terre'Blanche, MM Van der Walt, LJ Legoabe Bioorganic Chemistry 74, 251-259, 2017 | 21 | 2017 |
| The adenosine receptor affinities and monoamine oxidase B inhibitory properties of sulfanylphthalimide analogues MM Van der Walt, G Terre’Blanche, A Petzer, JP Petzer Bioorganic chemistry 59, 117-123, 2015 | 20 | 2015 |
| Imidazo [1, 2-α] pyridines possess adenosine A1 receptor affinity for the potential treatment of cognition in neurological disorders R Lefin, MM Van der Walt, PJ Milne, G Terre'Blanche Bioorganic & Medicinal Chemistry Letters 27 (17), 3963-3967, 2017 | 18 | 2017 |
| Selected C8 two-chain linkers enhance the adenosine A1/A2A receptor affinity and selectivity of caffeine MM Van der Walt, G Terre'Blanche European Journal of Medicinal Chemistry 125, 652-656, 2017 | 17 | 2017 |
| 2–Benzylidene–1–Indanone Analogues as Dual Adenosine A1/A2a receptor antagonists for the potential treatment of neurological conditions HDJ van Rensburg, LJ Legoabe, G Terre’Blanche, MM Van der Walt Drug research 69 (07), 382-391, 2019 | 16 | 2019 |
| Methoxy substituted 2-benzylidene-1-indanone derivatives as A 1 and/or A 2A AR antagonists for the potential treatment of neurological conditions HDJ van Rensburg, LJ Legoabe, G Terre'Blanche, MM Van der Walt Medchemcomm 10 (2), 300-309, 2019 | 15 | 2019 |
| Investigating the potential neuroprotective effects of statins on DNA damage in mouse striatum TN Coetsee, PJ Pretorius, G Terre’Blanche, JJ Bergh Food and chemical toxicology 46 (9), 3186-3192, 2008 | 15 | 2008 |
| Benzyloxynitrostyrene analogues–A novel class of selective and highly potent inhibitors of monoamine oxidase B MM Van der Walt, G Terre’Blanche, JP Petzer, A Petzer European journal of medicinal chemistry 125, 1193-1199, 2017 | 14 | 2017 |
