| 5-Substituted 2-benzylidene-1-tetralone analogues as A1 and/or A2A antagonists for the potential treatment of neurological conditions HDJ van Rensburg, G Terre'Blanche, MM Van der Walt, LJ Legoabe Bioorganic Chemistry 74, 251-259, 2017 | 21 | 2017 |
| 2–Benzylidene–1–Indanone Analogues as Dual Adenosine A1/A2a receptor antagonists for the potential treatment of neurological conditions HDJ van Rensburg, LJ Legoabe, G Terre’Blanche, MM Van der Walt Drug research 69 (07), 382-391, 2019 | 16 | 2019 |
| Methoxy substituted 2-benzylidene-1-indanone derivatives as A 1 and/or A 2A AR antagonists for the potential treatment of neurological conditions HDJ van Rensburg, LJ Legoabe, G Terre'Blanche, MM Van der Walt Medchemcomm 10 (2), 300-309, 2019 | 15 | 2019 |
| Synthesis and evaluation of methoxy substituted 2-benzoyl-1-benzofuran derivatives as lead compounds for the development adenosine A1 and/or A2A receptor antagonists HDJ van Rensburg, LJ Legoabe, G Terre'Blanche, J Aucamp Bioorganic Chemistry 94, 103459, 2020 | 10 | 2020 |
| C3 amino-substituted chalcone derivative with selective adenosine rA1 receptor affinity in the micromolar range HD Janse van Rensburg, LJ Legoabe, G Terre’Blanche Chemical Papers 75, 1581-1605, 2021 | 8 | 2021 |
| Synthesis and structure activity relationships of chalcone based benzocycloalkanone derivatives as adenosine A1 and/or A2A receptor antagonists HDJ van Rensburg, LJ Legoabe, G Terre’Blanche Drug Research 70 (06), 243-256, 2020 | 7 | 2020 |
| Synthesis and in vitro antileishmanial activity of alkylene-linked nitrofurantoin-triazole hybrids NH Zuma, J Aucamp, HDJ van Rensburg, DND David European Journal of Medicinal Chemistry 246, 115012, 2023 | 5 | 2023 |
| Exploration of chalcones and related heterocycle compounds as ligands of adenosine receptors: therapeutics development C Matthee, G Terre’Blanche, LJ Legoabe, HD Janse van Rensburg Molecular Diversity, 1-43, 2022 | 5 | 2022 |
| Design, synthesis and evaluation of amino-3,5-dicyanopyridines and thieno[2,3-b]pyridines as ligands of adenosine A1 receptors for the potential treatment of … G Nkomba, G Terre’Blanche, HD Janse van Rensburg, LJ Legoabe Medicinal Chemistry Research 31 (8), 1277-1297, 2022 | 4 | 2022 |
| Chalcone‐inspired rA1/A2A adenosine receptor ligands: Ring closure as an alternative to a reactive substructure C Matthee, G Terre’Blanche, HD Janse van Rensburg, J Aucamp, ... Chemical Biology & Drug Design 99 (3), 416-437, 2022 | 3 | 2022 |
| Striatal adenosine A2A receptor involvement in normal and large nest building deer mice: Perspectives on compulsivity and anxiety D Saaiman, L Brand, G de Brouwer, HJ van Rensburg, G Terre’Blanche, ... Behavioural Brain Research 449, 114492, 2023 | 2 | 2023 |
| New fused pyrroles with rA1/A2A antagonistic activity as potential therapeutics for neurodegenerative disorders NJ van Vuuren, HDJ van Rensburg, G Terre’Blanche, LJ Legoabe Molecular Diversity 26 (4), 2211-2220, 2022 | 2 | 2022 |
| Exploration of ethylene glycol linked nitrofurantoin derivatives against Leishmania: Synthesis and in vitro activity K Ndlovu, C Kannigadu, J Aucamp, HDJ Van Rensburg, DD N'Da Archiv der Pharmazie 356 (5), 2200529, 2023 | 1 | 2023 |
| Design, synthesis, electrochemistry and anti-trypanosomatid hit/lead identification of nitrofuranylazines M Saayman, C Kannigadu, J Aucamp, HDJ van Rensburg, C Joseph, ... RSC Medicinal Chemistry 14 (10), 2012-2029, 2023 | 1 | 2023 |
| Prophylactic activity of orally administered dry-heat-sterilized Acremonium egyptiacum against Trypanosoma congolense-induced animal African trypanosomosis A Yamazaki, Y Tanaka, K Watanabe, M Sato, S Kawazu, K Kita, N Inoue, ... Acta Tropica 254, 107185, 2024 | | 2024 |
| In vitro trypanocidal potency and in vivo treatment efficacy of oligomeric ethylene glycol-tethered nitrofurantoin derivatives HDJ van Rensburg, DND David, K Suganuma European Journal of Pharmaceutical Sciences 192, 106668, 2024 | | 2024 |
| Evaluation of chemical constituents of Rooibos (Aspalathus linearis) and Honeybush (Cyclopia intermedia) as adenosine A1/A2A receptor ligands L Gouws, HD Janse van Rensburg, G Terre’Blanche, MM Van der Walt Medicinal Chemistry Research 32 (12), 2535-2548, 2023 | | 2023 |
| In Vitro and In Vivo Trypanocidal Efficacy of Nitrofuryl- and Nitrothienylazines HD Janse van Rensburg, DD N’Da, K Suganuma ACS omega 8 (45), 43088-43098, 2023 | | 2023 |
| Preliminary Screening of South African Plants for Binding Affinity to the Serotonin Reuptake Transporter and Adenosine A1/A2A Receptors A Mnqika, AO Aremu, HD Janse van Rensburg, M Lekhooa Scientia Pharmaceutica 91 (3), 41, 2023 | | 2023 |
| On the basis of sex: male vs. female rat adenosine A1/A2A receptor affinity HD Janse van Rensburg, G Terre’Blanche, MM Van der Walt BMC Research Notes 16 (1), 165, 2023 | | 2023 |
Gisella Terre'BlancheSchool of Pharmacy, North-West University, Potchefstroom campusVerified email at nwu.ac.za
